Example: confidence

導美睡 7.5 Dormicum - roche.com.tw

Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 1 1018-DOR-01 Dormicum roche Film-Coated tablets mg 017577 Midazolam 1. / Dormicum benzodiazepines ATC code: N05CD08. / midazolam maleate midazolam midazolam maleate anhydrous lactose microcrystalline cellulose pregelatinized starch magnesium stearate titanium dioxide talc hypromellose ( Dormicum anhydrous lactose Lactose monohydrate [ ]) 2. (14 ) Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 2

Product Information Ro 21-3981 Dormicum, tablets 1 Product information Chinese

Tags:

  Tablets, Roche, Dormicum

Information

Domain:

Source:

Link to this page:

Please notify us if you found a problem with this document:

Other abuse

Advertisement

Transcription of 導美睡 7.5 Dormicum - roche.com.tw

1 Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 1 1018-DOR-01 Dormicum roche Film-Coated tablets mg 017577 Midazolam 1. / Dormicum benzodiazepines ATC code: N05CD08. / midazolam maleate midazolam midazolam maleate anhydrous lactose microcrystalline cellulose pregelatinized starch magnesium stearate titanium dioxide talc hypromellose ( Dormicum anhydrous lactose Lactose monohydrate [ ]) 2. (14 ) Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 2 2 Dormicum 15 Dormicum 30-60 / / Dormicum 7-8 ( )

2 Midazolam 1 -hydroxymidazolam glucuronide - - - - - benzodiazepines - - ketoconazole itraconazole voriconazole HIV ritonavir (boosted) ( ) Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 3 benzodiazepines benzodiazepines ( ) 2 Dormicum ( ) Dormicum ( ) Dormicum (anterograde amnesia) 7-8 ( ) Dormicum 15 7-8 (Psychiatric and paradoxical reactions) benzodiazepines / midazolam - Dormicum ( )

3 Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 4 Benzodiazepines Benzodiazepines / Dormicum / Dormicum / ( ) opioid Benzodiazepine opioid profound sedation Dormicum . CYP3A Midazolam CYP3A ( ) Lapp - Dormicum / Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 5 ( [ ])

4 ( ) - (DDI)( [ ]) midazolam P450 3A (CYP3A) CYP3A midazolam CYP3A midazolam CYP3A midazolam CYP3A CYP3A ( [mechanism based inhibition]) midazolam CYP3A clarithromycin erythromycin HIV verapamil diltiazem ethinylestradiol/norgestrel( ) midazolam CYP3A CYP3A midazolam Midazolam 10 3 ketoconazole itraconazole voriconazole HIV ritonavir (boosted) midazolam CYP3A ( )

5 Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 6 Midazolam 5 10 3 Midazolam 2 5 2 3 fluconazole clarithromycin telithromycin erythromycin diltiazem verapamil nefazodone aprepitant tabimoreline midazolam CYP3A midazolam ( [ ]) Midazolam 2 2 posaconazole roxithromycin cimetidine ranitidine fluvoxamine bicalutamide propiverine grapefruit juice echinacea purpurea goldenseal midazolam CYP3A midazolam CYP3A midazolam CYP3A midazolam CYP3A CYP3A rifampicin carbamazepine phenytoin efavirenz St John s wort - (DDI) midazolam / / / ( ) benzodiazepines (barbiturates) propofol ketamine etomidate Midazolam (MAC) midazolam ( )

6 Midazolam ( ( )) ( ) / ( AchE physostigmine) midazolam 250 midazolam Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 7 midazolam benzodiazepines midazolam benzodiazepines benzodiazepines midazolam Dormicum ( ).

7 Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 8 benzodiazepines (Psychiatric and paradoxical reactions) benzodiazepines benzodiazepines ( ) ( [ ]) : ( [ ]) : : : : : benzodiazepine ( ).

8 Benzodiazepines Dormicum Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 9 benzodiazepine Benzodiazepines ( ) 1-2 / flumazenil ( ) benzodiazepine flumazenil ( 1 ) Flumazenil ( ) flumazenil ( ) 3.

9 Dormicum / Dormicum benzodiazepines Dormicum gamma-aminobutyric acid(GABAA) benzodiazepines GABAA GABA Midazolam midazolam 30-70% midazolam Product Information Ro 21-3981 Dormicum , tablets Product information Chinese 10 Dormicum 15 1 70-120ng/ midazolam 5-20 midazolam 1-2 / 96-98% Midazolam midazolam midazolam Midazolam 1% Midazolam cytochrome P450 CYP3A CYP3A4 CYP3A5 midazolam 1 -hydroxymidazolam ( -hydroxymidazolam)

10 4-hydroxymidazolam 1 -hydroxymidazolam 60-80% glucuronic acid 1 -hydroxymidazolam conjugate 1 -hydroxymidazolam 30-50% 1 -hydroxymidazolam midazolam ( 34%) midazolam midazolam midazolam midazolam 1 -hydroxymidazolam 1 60 midazolam midazolam Product Information Ro 21-3981