Transcription of 【組成・性状】 - info.pmda.go.jp
1 2012 12 2 . 2012 8 8 7 2 3 9 9. 2. 5mg 22400 AMX01149000.. 5 mg 22400 AMX01150000. 2012 12 . 2012 12 .. 1 .. 2 5mg .. 5 mg 1 . 2 .. 2 5mg 5 mg . 2 65mg 5 29mg .. 2 5mg 5 mg .. 6000 . 3 . 2 .. mg 1) .. 82 5. A S T G O T A L T G P T . 2 5mg -GTP .. 113 . 5 mg . 2) .. 1 15mg A L T G P T A S T G O T A L P .. -GTP . 3 .. 1 . 1) 4 .. 2 .. 2) . 1 7 5mg .. 1 . 5 2 3 . 1) 2 5mg . 5 mg .. 2) .. 6 .. 7 . , - 100 . PTP PTP .. PTP . 99 5 .. , - 1 20 .. 8 .. 100 330 30 100mg/kg/ . Mosapride Citrate Hydrate 104 92 . 4-Amino-5-chloro-2-ethoxy.
2 - 2 - . 4- 4-fluorobenzyl morpholin-2-yl . methyl benzamide . monocitrate dihydrate C21H25 ClFN3O3 C6H8O7 2H2O.. 650 05. 1 1 , 2 . 5 mg . 1 . 5 mg . AUC . Cmax 90 . log 0. 8 log 1. 25 .. 2 5mg .. 5 mg .. 4 , 5 . 40 75 6 . 2 5mg . 5 mg 3 .. 2 5mg . PTP 100 10 10 . 5 mg . PTP 100 10 10 . 420 21 20 . 5 mg 500 10 50 . 1000 .. AUCt Cmax Tmax T1/2. ng hr/mL ng/mL hr hr 1 5 mg .. 23 47 5 17 6 22 5 9 9 0 8 0 6 1 88 0 27. 5 mg 2 2 5mg .. 23 48 5 18 1 21 7 9 4 0 9 0 3 1 85 0 26. 5 mg 3 2 5mg 5 mg . Mean S D . AUC Cmax 4 2 5mg.
3 5 5 mg .. 2 .. Meiji Seika . 104-8002 2-4-16. 0120 093-396 03 3273-3539. FAX 03 3272-2438.. 3 B-MOP.
